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24 April 2007 Poster Session 1: 17:35 - 19:00
P001 A fine line between agonism and antagonism at chemokine receptor CCR3
E. Wise, C. Duchesnes, P. Da Fonseca, R. Allen, T. Williams and J. Pease
P002 Visualization of differential conformational changes within the 3rd intracellular loop of the a2a-adrenergic receptor for full and partial agonists by optical recording in living cells
A. Zürn, U. Zabel, J.-P. Vilardaga, M.J. Lohse and C. Hoffmann
P003 Neurotensin Receptor 1: E.coli expression, purification, characterization and biophysical studies
P. Harding, J. Koeppe, H. Attrill, S. Ross, A. Kapanedis and A. Watts
P004 Differential orexin receptor internalization and recycling kinetics attributed to distinct b-arrestin interactions
K.D.G. Pfleger, M.B. Dalrymple, R.M. Seeber and K.A. Eidne
P005 A novel b-arrestin assay for monitoring GPCR activation
A. Fowler
P006 The role of Helix 8 residues of the V1b vasopressin receptor in receptor function
A. Baker and M. Wheatley
P007 A genetic approach to study the function of latrophilin in C. elegans
A.A. Adenle, D. de Pomerai and D.R. Bell
P008 Functional implications of family B receptor and ligand gene paralogues in teleosts
J. Cardoso, F. Vieira, A. Gomes and D. Power
P009 The agonist binding site of the V1b receptor
Y. Cashmore and M. Wheatley
P010 Just an extracellular loop? ECL 2 is critical for GPCR function
M. Conner and M. Wheatley
P011 Development of a non-imaging, homogenous assay format for analysis of arrestin recruitment as a detection method for generic GPCR screening
T. Wehrman, K. Peng, D. Bassoni, A. Fowler and K. Olsen
P012 Vasopressin/oxytocin receptors… and love: towards rational design of a central non peptide agonist
M.-C. Frantz, H. Chabane, J. Rodrigo, D. Rognan, T. Durroux, B. Mouillac, J.-P. Humbert, J. Haïech and M. Hibert
P013 Agonist-dependent consequences of proline to alanine substitution in the transmembrane helices of the calcitonin receptor
R.J. Bailey and D.L. Hay
P014 [3H]Org 43553, the first small molecule radioligand at the human luteinizing hormone (LH) receptor.
L.H. Heitman, J. Oosterom, C.M. Timmers, P. Wiegerinck and A.P. IJzerman
P015 Are functionally important contacts established between the N-terminus and extracellular loop-1 of the V1a vasopressin receptor?
R. Kendrick, J. Simms, D.L. Wootten, J. Trim and M. Wheatley
P016 Inverse agonist exposure enhances ligand binding and G protein activation of the human MT1 melatonin receptor, but leads to receptor down-regulation
T. Kokkola, M. Vaittinen and J.T. Laitinen
P017 Simulations of positive and negative cooperativity based on model of tandemly arranged ligand binding sites in receptor dimer. Case of melanocortin 4 receptor subtype
S. Kopanchuk, S. Veiksina, J.E.S. Wikberg and A. Rinken
P018 Determining the ligand binding selectivity for the parathyroid hormone receptors
R. Mann, M. Wigglesworth and D. Donnelly
P019 Ligand binding and activation of chemokine receptor CXCR6
S.J. Petit, N. Chayen and J.E. Pease
P020 The role of second extracellular loop of the CGRP receptor in ligand recognition
A.C. Conner, A. Ioannidou, J. Simms, J. Barwell, M. Wheatley and D.R. Poyner
P021 The role of the N-terminus of the CL receptor in binding CGRP
J. Simms, A.C. Conner, K. Mahmoud, M. Wheatley and D.R. Poyner
P022 Identification of residues required for high affinity CGRP binding on RAMP1 by means of RAMP1-RAMP3 chimeras
J. Simms, M. Wheatley and D.R. Poyner
P023 Pharmacological characterisation of the rat corticotropin-releasing factor (CRF) type 2b receptor (CRF-R2b) in transfected CHO cells and identification of a novel splice variant (CRF2del)
J.M.-N. Rainard, S.E. Mireylees and M.G. Darlison
P024 Expression of mammalian GPCRs in C. elegans generates novel behavioural responses to human ligands
M.S. Teng, M.P.J. Dekkers, B.-L. Ng, S. Rademakers, G. Jansen, A. Fraser and J. McCafferty
P025 Novel highly selective low-molecular radioligand for melanocortin-4 receptor: [125I]THIQ
S. Veiksina, S. Kopanchuk, F. Mutulis, J.E.S. Wikberg and A. Rinken
P026 Dopaminergic regulation of adenylyl cyclase activity in rat striatal homogenate
A. Vonk, R. Reinart and A. Rinken
P027 Expression and function of the GIPR in SGBS cells
R. Weaver, A. Balmforth and D. Donnelly
P028 Elucidating direct binding contacts between vasopressin and the V1a vasopressin receptor
D.L. Wootten, J. Simms, J. Trim and M. Wheatley
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